![cover image](https://wikiwandv2-19431.kxcdn.com/_next/image?url=https://upload.wikimedia.org/wikipedia/commons/thumb/a/a0/Osemozotan.svg/640px-Osemozotan.svg.png&w=640&q=50)
Osemozotan
Pharmaceutical drug / From Wikipedia, the free encyclopedia
Dear Wikiwand AI, let's keep it short by simply answering these key questions:
Can you list the top facts and stats about Osemozotan?
Summarize this article for a 10 year old
Osemozotan (MKC-242) is a selective 5-HT1A receptor agonist with some functional selectivity, acting as a full agonist at presynaptic and a partial agonist at postsynaptic 5-HT1A receptors.[1] 5-HT1A receptor stimulation influences the release of various neurotransmitters including serotonin, dopamine, norepinephrine, and acetylcholine.[2] 5-HT1A receptors are inhibitory G protein-coupled receptor.[3]
![]() | |
Legal status | |
---|---|
Legal status |
|
Identifiers | |
| |
CAS Number |
|
PubChem CID | |
ChemSpider |
|
UNII |
|
CompTox Dashboard (EPA) | |
Chemical and physical data | |
Formula | C20H23NO4 |
Molar mass | 341.407 g·mol−1 |
3D model (JSmol) | |
| |
| |
![]() ![]() |
Osemozotan has been shown to have antidepressant, anxiolytic, antiobsessional, serenic, and analgesic effects through animal studies.[4][5][6][2] It is used to investigate the role of 5-HT1A receptors in modulating the release of dopamine and serotonin in the brain[7][8] and their involvement in addiction to stimulants such as cocaine and methamphetamine.[9][10][11][12][13]