4-氟派醋甲酯 (4-Fluoromethylphenidate),又稱4-FMPH和4F-MPH,是一種興奮劑,與哌醋甲酯相比,是一種效力更強的多巴胺再攝取抑制劑。[2][3][4]
Quick Facts 法律規範狀態, 法律規範 ...
4-氟派醋甲酯 |
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法律規範 |
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Methyl 2-(4-fluorophenyl)-2-(piperidin-2-yl)acetate
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CAS號 | 1354631-33-6 Y |
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PubChem CID | |
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ChemSpider | |
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UNII | |
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化學式 | C14H18FNO2 |
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摩爾質量 | 251.30 g·mol−1 |
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3D模型(JSmol) | |
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熔點 | 222.0[1] °C(431.6 °F) |
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FC1=CC=C(C=C1)C(C(=O)OC)C2CCCCN2
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InChI=1S/C14H18FNO2/c1-18-14(17)13(12-4-2-3-9-16-12)10-5-7-11(15)8-6-10/h5-8,12-13,16H,2-4,9H2,1H3 Key:XISBAJBPDVRSPG-UHFFFAOYSA-N
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Misra M, Shi Q, Ye X, Gruszecka-Kowalik E, Bu W, Liu Z, et al. Quantitative structure-activity relationship studies of threo-methylphenidate analogs. Bioorganic & Medicinal Chemistry. October 2010, 18 (20): 7221–38. PMID 20846865. doi:10.1016/j.bmc.2010.08.034.
Singh S. Chemistry, design, and structure-activity relationship of cocaine antagonists. Chemical Reviews. March 2000, 100 (3): 925–1024. PMID 11749256. doi:10.1021/cr9700538.