Pethidine intermediate A is a four-phenylpiperidine derivative that is a precursor to the opioid analgesic drug pethidine (meperidine). It is not known to have any analgesic activity in its own right, however other derivatives of pethidine with a 4-cyano group in place of the carboxylate ethyl ester have been found to be active,[2] so pethidine intermediate A might also show opioid effects. It is scheduled by UN Single Convention on Narcotic Drugs. It is a Schedule II Narcotic controlled substance in the United States and has an ACSCN of 9232. The 2014 annual manufacturing quota was 6 grammes (as an end product, presumably for research use).[3]
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| Routes of administration | N/A |
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| ECHA InfoCard | 100.020.771 |
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| Formula | C13H16N2 |
| Molar mass | 200.285 g·mol−1 |
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See also
- Moramide intermediate
- Methadone intermediate
- Pethidine intermediate B (norpethidine)
- Pethidine intermediate C (pethidinic acid)
References
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